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Author: Mei-Ling Chen, Gordon L. Amidon, Leslie Z. Benet, Hans Lennernas, Lawrence X. Yu
Keywords: BCS,BDDCS,biopharmaceutics classification system,biopharmaceutics drug disposition classification system,drug metabolism,drug permeability Summary: biopharmaceutics classification
biopharmaceutics drug disposition classification system The BCS (Biopharmaceutics Classification System), based
Pharmaceutical Research; Vol. 28 Number 7, Jul 2011;Published Date:06/30/2011; DOI: 10.1007/s11095-011-0438-1
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Author: Akash Khandelwal, Praveen M. Bahadduri, Cheng Chang, James E. Polli, Peter W. Swaan, Sean Ekins
Keywords: BCS,BDDCS,random forest,recursive partitioning,support vector machine Summary: Computational Models to Assign Biopharmaceutics Drug Disposition
BCS, Biopharmaceutics Classification System; A training set of 165 drugs for computational model
Pharmaceutical Research; Vol. 24 Number 12, Dec 2007;Published Date:11/30/2007; DOI: 10.1007/s11095-007-9435-9
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Author: M. Sherry Ku
Keywords: biopharmaceutics classification,decision tree,formulation,polymorphism,salt Summary: The Biopharmaceutics Classification System (BCS) is not only a useful tool for obtaining
biopharmaceutics classification; decision tree; formulation; polymorphism; salt. in pharmaceutical companies to utilize computational chem-
The AAPS Journal; Vol. 10 Number 1, Mar 2008;Published Date:02/29/2008; DOI: 10.1208/s12248-008-9020-0
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Author: Vincent H. L. Lee
Summary: Computational biopharmaceutics, proteomics, and
Pharmaceutical Research; Vol. 19 Number 8, Aug 2002;Published Date:07/31/2002; DOI: 10.1023/A:1020127516809
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Author: Peter W. Swaan
Summary: computational and systems biology of drug ADME/Tox will
biopharmaceutics.
Pharmaceutical Research; Vol. 26 Number 3, Mar 2009;Published Date:02/28/2009; DOI: 10.1007/s11095-009-9836-z
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Author: Arik Dahan, Jonathan M. Miller, Gordon L. Amidon
Keywords: BA/BE,biopharmaceutics classification system,biowaiver,intestinal absorption,molecular biopharmaceutics,oral drug product Summary: The Biopharmaceutics Classification System (BCS) categorizes drugs into one of four
BA/BE; biopharmaceutics classification system; biowaiver; intestinal absorption; molecular biopharmaceutics; oral drug product.
The AAPS Journal; Vol. 11 Number 4, Dec 2009;Published Date:11/30/2009; DOI: 10.1208/s12248-009-9144-x
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Author: Filippos Kesisoglou, Amitava Mitra
Keywords: bioavailability enhancement,nanocrystals,nanoparticles,nanosizing,nanosuspensions Summary: oral absorption of Biopharmaceutics Classification System class II and IV compounds. based on the Biopharmaceutics Classification System (BCS) (1) to achieve 1 Biopharmaceutics, Product Value Enhancement, Pharmaceutical Sciences and Clinica
The AAPS Journal; Vol. 14 Number 4, Dec 2012;Published Date:11/30/2012; DOI: 10.1208/s12248-012-9383-0
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Author: Caroline A. Larregieu, Leslie Z. Benet
Keywords: Biopharmaceutics Classification System (BCS),biowaiver,Caco-2 cells,Food and Drug Administration (FDA),human intestinal permeability,in silico modeling,in vitro screening Summary: Biopharmaceutics Classification System (BCS); biowaiver; Caco-2 cells; Food and Drug Administration inception of the Biopharmaceutics Classification System (BCS), which originally demonstrated a rela
The AAPS Journal; Vol. 15 Number 2, Apr 2013;Published Date:03/31/2013; DOI: 10.1208/s12248-013-9456-8
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